| Patent Number |
Title Of Patent |
Date Issued |
| 6432948 |
USE OF 7-(2-OXA-5,8-DIAZABICYLCO[4.3.0]NON-8-YL)-QUINOLONE CARBOXYLIC ACID AND NAPHTHYRIDON CARB |
August 13, 2002 |
| The invention relates to the use of quinolone- and naphthyridonecarboxylic acid derivatives, which are substituted in the 7-position by a 2-oxa-5,8-diazabicyclo[4.3.0]-non-8-yl) radical, and their pharmaceutically utilizable hydrates and/or salts for the therapy of Helicobacter pylor |
| 6288081 |
Use of 7-(1-aminomethyl-2-oxa-7-aza-bicyclo[3.3.0]oct-7-yl)-quinolone carboxylic acid and naphth |
September 11, 2001 |
| The invention relates to the use of quinolone- and naphthyridonecarboxylic acid derivatives which are substituted in position 7 by a 1-aminomethyl-2-oxa-7-azabicyclo[3.3.0]oct-7-yl radical, and of their salts for the therapy of Helicobacter pylori infections and associated gastroduod |
| 6204272 |
Use of aminothiazoles for treating wounds and skin |
March 20, 2001 |
| The invention relates to the use of substituted 2-aminothiazoles for promoting wound healing. |
| 6133260 |
Use of 7-(2-oxa-5,8-diazabicyclo[4.3.0]non-8-yl)-quinolone carboxylic acid and naphthyridon carb |
October 17, 2000 |
| The invention relates to the use of quinolone- and naphthyridonecarboxylic acid derivatives which are substituted in the 7-position by a 2-oxa-5,8-diazabicyclo[4.3.0]-non-8-yl) radical, and their pharmaceutically utilizable hydrates and/or salts for the therapy of Helicobacter pylori |
| 6069160 |
Heteroatom-containing benzocyclopentane-oxazolidinones |
May 30, 2000 |
| The invention relates to heteroatom-containing benzocyclopentaneoxazolidinones, to processes for their preparation and their use as medicaments, especially as antibacterial medicaments. |
| 6034055 |
Glycosyl-amides of 2-aminoacylamino-2-deoxy-sugars |
March 7, 2000 |
| The present invention relates to (2-aminoacylamino-2-deoxy-glycosyl)-amides, which are substituted on the nitrogen atom of the amino acid, of the general formula (I) ##STR1## in which the substituents have the meaning given in the description, to processes for their preparation a |
| 5905071 |
Glycosylamides of 2-aminoacylamino-2-deoxy sugars |
May 18, 1999 |
| The present invention relates to (2-aminoacylamino-2-deoxy-glycosyl)-amides, which are substituted on the nitrogen atom of the amino acid, of the general formula (I) ##STR1## in which the substituents have the meaning given in the description, to processes for their preparation a |
| 5843967 |
6-membered nitrogen-containing heteroaryl-oxazolidinones |
December 1, 1998 |
| The invention relates to 6-membered nitrogen-containing heteroaryloxazolidinones, processes for their preparation and their use as medicaments, in particular as antibacterial medicaments. |
| 5698574 |
5-membered heteroaryl-oxazolidinones |
December 16, 1997 |
| The present invention relates to 5-membered heteroaryl-oxazolidinones, to processes for their preparation and to their use as medicaments, in particular as antibacterial medicaments. |
| 5684023 |
Benzofuranyl -and benzothienyloxazolidinones |
November 4, 1997 |
| The present invention relates to benzofuranyl- and benzothienyloxazolidinones, processes for their preparation and their use as medicaments, in particular as antibacterial medicaments. |
| 5627181 |
6-membered nitrogen-containing heteroaryl-oxazolidinones |
May 6, 1997 |
| The invention relates to 6-membered nitrogen-containing heteroaryloxazolidinones, processes for their preparation and their use as medicaments, in particular as antibacterial medicaments. |
| 5529998 |
Benzoxazolyl- and benzothiazolyloxazolidinones |
June 25, 1996 |
| The invention relates to benzoxazolyl- and benzothiazolyloxazolidinones, processes for their preparation and their use as medicaments, in particular as antibacterial medicaments. |
| 5350861 |
Substituted 3-aryl-pyrrolidine-2,4-diones |
September 27, 1994 |
| There are provided new substituted 3-aryl-pyrrolidine-2,4-diones of the formula ##STR1## in which X represents hydrogen, alkyl, halogen or alkoxy,Y represents hydrogen, alkyl, halogen, alkoxy or halogenoalkyl,Z represents alkyl, halogen or alkoxy,n represents a number from 0-3,R represen |
| 5330976 |
Antimycotic compositions of nikkomycin compounds and azole antimycotics |
July 19, 1994 |
| Nikkomycin compounds have been found to be orally or parenterally effective as anti-fungals in animals. They may be used alone or, preferably, in combination with azole antimycotics for a synergistic anti-fungal effect. |
| 5258394 |
1-trifluoromethyl-1-nitro-2-alkoxy-2-aryl-ethanes, their preparation and antimycotic agents cont |
November 2, 1993 |
| 1-Trifluoromethyl-1-nitro-2-alkoxy-2-aryl-ethanes of the formula ##STR1## in which R.sup.1 represents a straight-chain or branched alkyl radical andR.sup.2 represents an optionally substituted aryl or hetaryl radical,their preparation from an aldehyde of the formula R.sup.2 --CHO, an alcohol |
| 5194427 |
Antimycotic compositions of nikkomycin compounds and azole antimycotics |
March 16, 1993 |
| Nikkomycin compounds have been found to be orally or parenterally effective as anti-fungals in animals. They may be used alone or, preferably, in combination with azole antimycotics for a synergistic anti-fungal effect. |
| 5186737 |
Pesticidal 3-aryl-pyrrolidine-2,4-diones |
February 16, 1993 |
| Insecticidal, acaricidal, herbicidal and antimycotic 3-aryl-pyrrolidine-2,4-diones of the formula ##STR1## in which X represents alkyl, halogen or alkoxy,Y represents hydrogen, alkyl, halogen, alkoxy or halogenoalkyl,Z represents alkyl, halogen or alkoxy,n represents a number from 0-3,R |
| 5149795 |
Nikkomycin derivatives |
September 22, 1992 |
| The nikkomycin compound possessing antimycotic activity and having the following structure: ##STR1## |
| 5142092 |
Fluorine-containing acetophenones optionally halogenated on the CH.sub.3 -group and their precur |
August 25, 1992 |
| Fluorine-containing acetophenones, optionally halogenated on the CH.sub.3 group, of the formula ##STR1## in which X represents hydrogen, chlorine or bromine and the radicals R.sub.1 to R.sub.5 have the following meaning,a) R.sub.1 and R.sub.4 denote fluorine, R.sub.2 and R.sub.5 deno |
| 5142065 |
3-aryl-pyrrolidine-2,4-diones |
August 25, 1992 |
| An acylamino ester of the formula ##STR1## wherein X is C.sub.1-6 alkyl, or halogen,Y is hydrogen, C.sub.1-6 alkyl, halogen, or C.sub.1-3 halogenalkyl,Z is C.sub.1-6 alkyl, or halogen,n is 0 to 3,provided that when n is O,Y is not hydrogen, andR.sup.3 is C.sub.1-6 alkyl. |
| 5134126 |
Antimycotic compositions of nikkomycin compounds and azole antimycotics |
July 28, 1992 |
| Nikkomycin compounds have been found to be orally or parenterally effective as anti-fungals in animals. They may be used alone or, preferably, in combination with azole antimycotics for a synergistic anti-fungal effect. |
| 5104879 |
Antimycotically active substituted 2-aminothiazoles |
April 14, 1992 |
| Antimicotically active 2-aminothiazoles have been found having the formula ##STR1## in which R.sup.1 represents hydrogen or alkyl andR.sup.2 represents optionally substituted cyclohexyl or phenyl which is substituted by halogen, alkyl, halogenoalkyl, halogenoalkoxy, dioxyhalogenoalky |
| 5096889 |
Antimycotic compositions of nikkomycin compounds and azole antimycotics |
March 17, 1992 |
| Nikkomycin compounds have been found to be orally or parenterally effective as anti-fungals in animals. They may be used alone or, preferably, in combination with azole antimycotics for a synergistic anti-fungal effect. |
| 5091537 |
Intermediates for preparing 3-aryl-pyrrolidine-2,4-diones |
February 25, 1992 |
| A 3-aryl-pyrrolidine-2,4-dione (e) derivative of the formula (I) ##STR1## in which X represents alkyl, halogen and alkoxy,Y represents hydrogen, alkyl, halogen, alkoxy and halogenoalkyl,Z represents alkyl, halogen and alkoxy,m represents a number from 1-4,n represents a number from 0-3,R rep |
| 5091375 |
Nikkomycin derivatives |
February 25, 1992 |
| Nikkomycin derivatives have been found to be orally or parenterally effective as anti-fungals in animals. They may be used alone or, preferably, in combination with azole antimycotics for a synergistic anti-fungal effect. |
| 5045560 |
Pesticidal tautomers of 3-aryl-pyrrolidine-2,4-diones and use thereas |
September 3, 1991 |
| Insecticidal, acaricidal, herbicidal and antimycotic 3-aryl-pyrrolidine-2,4-diones of the formula ##STR1## in which X represents alkyl, halogen or alkoxy,Y represents hydrogen, alkyl, halogen, alkoxy or halogenoalkyl,Z represents alkyl, halogen or alkoxy,n represents a number from 0-3,R |
| 5019560 |
Method for treating fungal infections with nikkomycin derivatives |
May 28, 1991 |
| A method of treating a mammal infected with a dimorphic, highly chitinous fungi, the method comprising administering to the mammal therapeutically effective amounts of a nikkomycin derivative having the following structure: ##STR1## |
| 5011850 |
Substituted diazolylalkyl-carbinols, a process for their preparation and their use as antimycoti |
April 30, 1991 |
| The invention relates to compounds and their derivatives, said compounds being described herein as those of Formula (I). The compounds and compositions containing them are effective antimycotic agents and the invention includes methods for the use of said compounds and compositions. |
| 5006513 |
Antimycotic compositions of nikkomycin compounds and azole antimycotica |
April 9, 1991 |
| Nikkomycin compounds have been found to be orally or parenterally effective as anti-fungals in animals. They may be used alone or, preferably, in combination with azole antimycotics for a snyergistic anti-fungal effect. |
| 4985063 |
3-aryl-pyrrolidine-2,4-diones |
January 15, 1991 |
| A 3-aryl-pyrrolidine-2,4-dione (e) derivative of the formula (I) ##STR1## in which X represents alkyl, halogen and alkoxy,Y represents hydrogen, alkyl, halogen, alkoxy and halogenoalkyl,Z represents alkyl, halogen and alkoxy,m represents a number from 1-4,n represents a number from 0-3, R re |
| 4956370 |
Antimycotically active substituted 2-aminothiazoles |
September 11, 1990 |
| A 2-aminothiazole of the formula ##STR1## in which R.sup.1 represents hydrogen or alkyl andR.sup.2 represents a radical of the formula ##STR2## where R.sup.3, R.sup.4, R.sup.5 and R.sup.6 independently of one another in each case represent hydrogen, halogen, nitro, alkyl, alkoxy |
| 4914087 |
Nikkomycin derivatives, antimycotic compositions of nikkomycin derivatives and azole antimycotic |
April 3, 1990 |
| Nikkomycin derivatives have been found to be orally or parenterally effective as anti-fungals in animals. They may be used alone or, preferably, in combination with azole antimycotics for a synergistic anti-fungal effect. |
| 4894382 |
Substituted 1,3-diazolyl-2-propanols and their use as antimycotic agents |
January 16, 1990 |
| The invention provides substituted 1,3-diazolyl-2-propanols defined herein generically by formula (I), useful as antimycotic agents. Also included in the invention are methods for the procurement of said substituted 1,3-diazolyl-2-propanols, compositions containing said antimycotic c |
| 4879385 |
Substituted hydroxyalkyl-azoles and their use as antimycotics |
November 7, 1989 |
| The invention relates to substituted hydroxyalkylazoles defined herein by formula (I), which compounds are useful as antimycotic agents. Also included in the invention are compositions containing said compounds and methods for the use of said compounds and compositions. In addition, the |
| 4855283 |
Novel pharmaceutically active N-(2-aminoacylamido-2-deoxy-hexosyl)-amides, -carbamates and -urea |
August 8, 1989 |
| Compounds of the formula ##STR1## in which R.sup.1 denotes hydrogen or a saturated or singly or multiply unsaturated alkyl radical having up to 50 carbon atoms,X represents --CH.sub.2 --, --O-- or --NH--,R.sup.2 denotes hydrogen or a saturated or singly or multiply unsaturated alkyl |
| 4806559 |
Novel substituted hydroxyalkyl-azole antimycotic agents |
February 21, 1989 |
| An antimycotic agent, comprising a compound of the formula ##STR1## in which R.sup.1 is hydrogen, alkyl, optionally substituted phenyl or optionally substituted benzyl,R.sup.2 is hydrogen, alkyl, alkenyl, alkynyl, optionally substituted phenyl or optionally substituted benzyl,R.sup.3 |
| 4737488 |
Immune system-stimulating N-glycosylated ureas and carbamates |
April 12, 1988 |
| Compounds of the formula ##STR1## wherein R.sup.1 is hydrogen, an optionally substituted aromatic hydrocarbon radical, an aralkyl radical or an optionally substituted aliphatic hydrocarbon radical having up to 45 C atoms,R.sup.2 is an optionally substituted aromatic hydrocarbon radic |
| 4716152 |
Pharmaceutical use of substituted O-acylglycosides |
December 29, 1987 |
| Compounds of the formula ##STR1## in which X is hydrogen or the radical CH.sub.2 OR.sup.5,R.sup.2, R.sup.3, R.sup.4 and R.sup.5 each independently is hydrogen or the radical ##STR2## Y is oxygen, sulphur, NH or CH.sub.2, and R.sup.1 and R.sup.6 each independently is an option |
| 4683222 |
N-glycosylated carboxamide derivatives and their use for influencing the body's inherent defence |
July 28, 1987 |
| The invention relates to N-glycosylated carboxamide derivatives of Formula I which are useful for influencing the body's inherent defenses, e.g. for increasing immune system antibodies. Also included in the invention are compositions containing said N-glycosylated carboxamide derivative |
| 4631272 |
N-acylated 1-alkylamino-1-deoxy-ketose derivatives, a process for their preparation and their us |
December 23, 1986 |
| Compounds of the formula ##STR1## in which R.sup.1 represents hydrogen or an optionally substituted, straight-chain or branched alkyl or mono- or poly-unsaturated alkenyl radical with in each case up to 30 C atoms,X represents CH.sub.2, O, S or NR,whereinR denotes hydrogen or an alky |
| 4581453 |
Guanidinothiazole derivatives containing alkylene bridges, and their use for influencing lipid m |
April 8, 1986 |
| The invention relates to guanidinothiazol derivatives of Formula (I) as defined herein, said compounds being useful for influencing lipid metabolism, as antithombotic agents and as antimycotic agents. Also included in the invention are compositions containing said guanidinothiazol de |
| 4558139 |
Bafilomycin pesticides |
December 10, 1985 |
| Bafilomycins of the formula ##STR1## in which R.sup.1 is hydrogen or CH.sub.3, andR.sup.2 is hydrogen, or the group ##STR2## are produced by culturing certain streptomyces, e.g. Tu/ 1922, Tu/ 2437 and Tu/ 2599. Those wherein at least one of the OH groups is acylated are n |
| 4487776 |
Azolyl-phenoxy-tetrahydrofuran-2-ylidene-methanes, a process for their preparation, and antimicr |
December 11, 1984 |
| The invention relates to azolyl-phenoxy-tetrahydrofuran-2-ylidene-methanes defined herein under formula (I). Also included in the invention are compositions containing said compounds of formula (I) and methods for the use of such compounds and compositions as antimycotic agents. The |
