| Patent Number |
Title Of Patent |
Date Issued |
| RE35754 |
Cephem derivatives |
March 24, 1998 |
| Cephem derivatives of the general formula ##STR1## is which the R.sub.2 O group is in the syn-position, a process for their manufacture and pharmaceutical formulations which are active against bacterial infections and contain these compounds. |
| RE34865 |
Cephalosporin derivatives |
February 21, 1995 |
| Cephemcarboxylic acid esters of the general formula ##STR1## pharmaceutical preparations which are active against bacterial infections, which contain such cephem derivatives, a process for the preparation of the cephem derivatives and the pharmaceutical preparations, and also the |
| 6835724 |
Corticoid 17,21-dicarboxylic esters and corticosteroid 17-carboxylic ester 21-carbonic esters, p |
December 28, 2004 |
| Corticoid 17,21-dicarboxylic esters and corticosteroid 17-carboxylic ester 21-carbonic esters, processes for their preparation and pharmaceuticals containing these compoundsCorticoid 17,21-dicarboxylic esters and corticoid 17-carboxylic ester 21-carbonic esters of the formula I: ##ST |
| 5747484 |
Crystalline cepham acid addition salts and processes for their preparation |
May 5, 1998 |
| Novel crystalline cephem acid addition salts and processes for their preparationCompounds of the formula I ##STR1## in which n is equal to 1 or 2 andm is 0.4-2.6, and where X is the anion of a carboxylic acid, have antibacterial activity. |
| 5710146 |
Cephem derivatives and processes for their manufacture |
January 20, 1998 |
| Cephem derivatives of the general formula ##STR1## in which the R.sub.2 O group is in the syn-position, a process for their manufacture and pharmaceutical formulations which are active against bacterial infections and contain these compounds. |
| 5608093 |
Corticosteroid 17-alkyl carbonate 21-[0]-carboxylic and carbonic esters, and pharmaceuticals con |
March 4, 1997 |
| Corticoid 17-alkyl carbonate 21-carboxylic and carbonic esters of the formula I ##STR1## are described in which A is CHOH and CHCl, CH.sub.2, C.dbd.O or 9(11) double bond; Y is H, F or Cl; Z is H, F or CH.sub.3 ; R(1) is aryl or hetaryl; n and m are zero or 1; R(2) is alkyl or -- |
| 5565423 |
Cyclopeptides and their use as absorption promoters when applied to the mucosa |
October 15, 1996 |
| Cyclopeptides and their use as absorption promoters when applied to the mucosaThe invention relates to a compound of the formula I ##STR1## or a physiologically tolerated salt thereof, in which X is a basic L- or D-amino acid,Y is a neutral or basic L- or D-amino acid,Z is a neutral |
| 5409918 |
Crystalline cephem acid addition salts and process for their preparation |
April 25, 1995 |
| Crystalline cephem acid addition salts of the general formula II ##STR1## pharmaceutical preparations effective against bacterial infections which contain such cephem derivatives, processes for the preparation of the cephem derivatives and the pharmaceutical preparations, and the use |
| 5362721 |
Corticoid-17-alkyl-carbonates substituted in the 17-position, process for their preparation and |
November 8, 1994 |
| The disclosed invention includes corticoid-17-alkylcarbonates substituted in the 17-position, a process for their preparation and pharmaceuticals containing them. These corticoid-17-alkylcarbonates have the following formula I ##STR1## where A is CHOH in any desired steric arrang |
| 5306717 |
Cephalosporin derivatives |
April 26, 1994 |
| Cephalosporin derivatives of the general formula ##STR1## pharmaceutical preparations which are active against bacterial infections and contain such cephem derivatives, processes for the preparation of the cephem derivatives and the pharmaceutical preparations and the use of the |
| 5100887 |
Cephalosporin derivatives |
March 31, 1992 |
| Cephemcarboxylic acid esters of the general formula ##STR1## pharmaceutical preparations which are active against bacterial infections, which contain such cephem derivatives, a process for the preparation of the cephem derivatives and the pharmaceutical preparations, and also the |
| 5091382 |
Cephalosporin derivatives |
February 25, 1992 |
| Cephalosporin derivatives of the general formula ##STR1## pharmaceutical preparations active against bacterial infections which contain such cephalosporin derivatives, processes for the preparation of the cephalosporin derivatives, use of the cephalosporin derivatives for the pre |
| 5089490 |
Cephem derivatives |
February 18, 1992 |
| Cephem derivatives of the general formula ##STR1## in which the R.sub.2 O group is in the syn-position, a process for their manufacture and pharmaceutical formulations which are active against bacterial infections and contain these compounds. |
| 5071979 |
Cephalosporin derivatives |
December 10, 1991 |
| What are disclosed are anti-bacterially active cephalosporin compounds of the formula ##STR1## pharmaceutical preparations containing such compounds, methods of making the compounds, methods for combatting bacterial infections therewith, and intermediates for such compounds. |
| 5036063 |
Penem derivatives |
July 30, 1991 |
| Penem derivatives of the formula ##STR1## having R.sup.1 equal to 3-oxocyclobutyl and R.sup.2 equal to H or an ester-forming group, pharmaceutical preparations active against bacterial infections and which contain penem derivatives of this type, processes for the preparation of t |
| 4845087 |
Crystallized cephem-acid addition salts, and a process for the preparation thereof |
July 4, 1989 |
| Crystallized cephem-acid addition salts of the general formula ##STR1## pharmaceutical preparations which contain such cephem derivatives and are active against bacterial infections, a process for the preparation of the cephem derivatives and the pharmaceutical preparations, and the |
| 4762848 |
1,3-thiazoles and their use as immunomodulators |
August 9, 1988 |
| Heterocyclic sulfides of the general formula heterocycle-S-R, a process for their preparation and, in particular, their use for immunostimulation, immunorestoration and cytostatic treatment, and pharmaceutical agents, which contain a sulfide of this type, for these indications. |
| 4758556 |
Cephem derivatives |
July 19, 1988 |
| Cephem derivatives of the general formula ##STR1## in which the R.sub.2 O group is in the syn-position, a process for their manufacture and pharmaceutical formulations which are active against bacterial infections and contain these compounds. |
| 4701452 |
Use of cephem compounds as immunomodulators |
October 20, 1987 |
| The use of cephem compounds of the general formula I ##STR1## to increase the immunological responsiveness of mammals and formulations which contain an effective content of cephem compounds of the general formula I. |
| 4692516 |
Process for the manufacture of 3-pyridinium-methyl-cephalosporins |
September 8, 1987 |
| Process for the preparation of cephem compounds of the formula ##STR1## wherein R is optionally substituted aminothiazolyl or amino-1,2,4-thiadiazolyl, A is optionally substituted pyridinium, R.sup.1 is hydrogen or methoxy and R.sup.2 are special aliphatic substituents, by a nucl |
| 4667028 |
Process for the preparation of cephem compounds |
May 19, 1987 |
| Process for the preparation of cephem compounds of the formula ##STR1## |
| 4647556 |
Cephalosporin derivatives |
March 3, 1987 |
| The invention relates to cephem derivatives of the general formula I ##STR1## and their physiologically acceptable acid addition salts, to pharmaceutical formulations active against bacterial infections, to processes for preparing the compounds and formulations, and to the use of |
| 4624948 |
Crystalline modification of ceftazidim |
November 25, 1986 |
| Anhydrous crystalline (6R,7R)-7-[(Z)-2-(2-aminothiazol-4-yl)-2-(2-carboxyprop-2-oximino)acetamid o]-3-(1-pyridiniummethyl)-3-cephem-4-carboxylate and a process for its preparation, a pharmaceutical formulation which is active against bacterial infections and contains this compound and |
| 4609653 |
Crystalline cephem-acid addition salts and processes for their preparation |
September 2, 1986 |
| Crystalline cephem-acid addition salts of the formula ##STR1## and their hydrates, processes for the preparation of the acid addition salts, pharmaceutical products containing these compounds and processes for their preparation, and the use of the compounds for combating bacteria |
| 4603129 |
Cephalosporin derivatives |
July 29, 1986 |
| What are disclosed are cephalosporin compounds of the formula ##STR1## pharmaceutical preparations which are active against bacterial infections and in which these cephem compounds are present, process for the preparation of the cephem compounds and of the pharmaceutical preparat |
| 4593027 |
3-aryl-7-chloro-3,4-dihydroacridine-1,9(2H,10H)-dione 1-oximes and 1-hydrazone derivatives, thei |
June 3, 1986 |
| 3-Aryl-7-chloro-3,4-dihydroacridine-1,9(2H,10H)-dione 1-oximes and 1-hydrazone derivatives of the formula I ##STR1## and their physiologically tolerated acid addition and ammonium salts are described, as is a process for their preparation. The new compounds are chemotherapeutic a |
| 4590267 |
Crystalline disodium salt of cefodizim |
May 20, 1986 |
| A crystalline water soluble disodium salt of 7-.beta.-[2-(2-aminothiazol-4-yl)-2-syn-methoximinoacetamido]-3-(5-carboxy methyl-4-methyl-1,3-thiazol-2-ylthiomethyl)ceph-3-em-4-carboxylic acid (cefodizim), or an adduct or solvate thereof with water and/or an organic solvent. |
| 4470983 |
Cephalosporin derivatives |
September 11, 1984 |
| What are disclosed are cephalosporin compounds of the formula ##STR1## pharmaceutical preparations which are active against bacterial infections and in which these cephem compounds are present, process for the preparation of the cephem compounds and of the pharmaceutical preparat |
| 4454129 |
Cephem derivatives |
June 12, 1984 |
| What are disclosed are cephem compounds of the formula ##STR1## useful for combating bacterial infections, and methods of making and using the same. |
| 4399131 |
Cephem derivatives |
August 16, 1983 |
| What are disclosed are cephem compounds of the formula ##STR1## in which R.sub.1 denotes hydrogen, an optionally substituted alkyl, acyl, arylsulfonyl or alkylsulfonyl group or an amino-protective group which is known from peptide chemistry, R.sub.2 denotes hydrogen or an optionally |
| 4293550 |
Cephalosporin derivatives |
October 6, 1981 |
| Cephalosporin derivatives of the formula ##STR1## processes for their manufacture and their use for combating bacterial infections. |
| 4284627 |
Antimalarial compositions |
August 18, 1981 |
| Antimalarial compositions are disclosed containing as the active ingredient a mixture of a tetrahydroacridone of the general formula I ##STR1## in which R.sup.1 represents methyl, phenyl, p-chlorophenyl, m-chlorophenyl, p-fluorophenyl, p-trifluoromethylphenyl, o-trifluoromethylph |
| 4282220 |
Cephem derivatives |
August 4, 1981 |
| What is disclosed are cephalosporin compounds of the formula ##STR1## pharmaceutical preparations having an action against bacterial infections and containing such cephem compounds, a process for the manufacture of the cephem compounds and of pharmaceutical preparations containing th |
| 4278793 |
Cephem derivative |
July 14, 1981 |
| Cephem derivatives of the general formula ##STR1## in which the R.sub.2 O group is in the syn-position, a process for their manufacture and pharmaceutical formulations which are active against bacterial infections and contain these compounds. |
| 4260615 |
Antimalarial compositions |
April 7, 1981 |
| Antimalarial compositions are disclosed containing as the active ingredient a mixture of a tetrahydroacridone of the general formula I ##STR1## in which R.sup.1 represents methyl, phenyl, p-chlorophenyl, m-chlorophenyl, p-fluorophenyl, p-trifluoromethylphenyl, o-trifluoromethylph |
| 3993694 |
Tetracycline derivatives and process for preparing them |
November 23, 1976 |
| Antibacterially-active tetracyclines, substituted at the amide group, and physiologically-tolerable salts thereof, said tetracyclines having the formula ##SPC1##Methods of making the same; pharmaceutical compositions containing the same. |
| 3983173 |
2-Carboxamido-substituted tetracyclines and process for their manufacture |
September 28, 1976 |
| 2-Carboxamido-substituted tetracyclines of the general formula ##SPC1##A process for their preparation and compositions containing these compounds. |
| 3947449 |
Tetrahydroacridones having chemotherapeutic action and process for preparing them |
March 30, 1976 |
| Tetrahydroacridones and their salts with physiologically tolerated acids and bases and process for preparing them. The compounds have a valuable chemotherapeutic action and may be used as drugs against protozoan diseases. |
