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Inventor:
Norcross; Roger David
Address:
Olsberg, CH
No. of patents:
15
Patents:












Patent Number Title Of Patent Date Issued
8188139 Heterocyclic-substituted phenyl methanones May 29, 2012
The present invention relates to compounds of formula I ##STR00001## wherein R.sup.1, R.sup.2, and are defined in the specification and to pharmaceutically acceptable acid addition salts thereof.
8153679 Radiolabelled inhibitors of the glycine 1 transporter April 10, 2012
The present invention relates to novel radiolabelled inhibitors of formula I for the Glycine 1 transporter (GlyT1), useful for the labelling and diagnostic imaging of the glycine 1 transporter functionality. ##STR00001## wherein R.sup.1 is isopropoxy or 2,2,2-trifluoro-1-methyl-etho
7790763 Substituted phenyl methanone derivatives September 7, 2010
The present invention relates to compounds of formula I ##STR00001## wherein R.sup.1, R.sup.2, R.sup.3, n, and m, are as defined in the specification and to pharmaceutically acceptable acid addition salts thereof. These compounds are good inhibitors of the glycine transporter 1 (G
7728142 3-methanesulfonylquinolines as GABA.sub.B enhancers June 1, 2010
The present invention relates to compounds of formula I ##STR00001## wherein R.sup.1, R.sup.2 and R.sup.3 are as defined in the specification, which are active at the GABA.sub.B receptor and which can be used for the treatment of CNS disorders.
7576217 Quinolines as allosteric enhancers of the GABA.sub.B receptors August 18, 2009
The present invention relates to compounds of formula I ##STR00001## wherein R.sup.1 to R.sup.6 are as described herein, which compounds are active at the GABA.sub.B receptor and can be used for the preparation of medicaments useful in the treatment of CNS disorders comprising anxiety
7557114 Heterocyclic-substituted phenyl methanones July 7, 2009
The present invention relates to compounds of formula I ##STR00001## wherein R.sup.1 and R.sup.2 are defined in the specification and to pharmaceutically acceptable acid addition salts thereof. Compounds of the invention are GlyT-1 inhibitors and are useful for the treatment of CNS d
7504428 2-phenyl-3,3,3-trifluoro-2-hydroxy-propionic acid derivatives March 17, 2009
The present invention a method of treating anxiety by administering compounds that are active on the GABA.sub.B receptor, having formula I: ##STR00001## wherein R.sup.1, R.sup.2, R.sup.3, R.sup.4, R.sup.5 and R.sup.6 are as defined in the specification and claims.
7485637 Benzoyl-tetrahydropiperidine derivatives February 3, 2009
The present invention relates to compounds of formula I ##STR00001## wherein R.sup.1, R.sup.2, and Ar; are as defined in the specification. The invention also provides pharmaceutically acceptable acid addition salts thereof and methods for the treatment of neurological and neuropsych
7442710 Substituted phenyl methanones October 28, 2008
The present invention relates to compounds of general formula IA or IB ##STR00001## wherein X.sup.1 and X.sup.2 are each independently N or C--R'' and R.sup.1, R.sup.2,R.sup.3, R.sup.4, R.sup.5, and R.sup.6 are as defined in the specification and to pharmaceutically acceptable acid
7429585 Phenyl-piperazine methanone derivatives, substituted by heterocyclic groups September 30, 2008
The present invention relates to compounds of the general formula IC ##STR00001## wherein R.sup.2, R', R'', R.sup.3, R.sup.6, X.sup.1 and X.sup.1' are as defined herein and pharmaceutically active acid addition salts thereof. Compounds of the invention are useful for the treatment of
7396853 2-phenyl-3,3,3-trifluoro-2-hydroxy-propionic acid derivatives July 8, 2008
The present invention relates to compounds of formula I: ##STR00001## wherein R.sup.1, R.sup.2, R.sup.3, R.sup.4, R.sup.5 and R.sup.6 are as defined in the specification and claims, which compounds are active on the GABA.sub.B receptor and are useful in the control or prevention of C
7390903 Thieno-pyridine derivatives as allosteric enhancers of the GABA.sub.B receptors June 24, 2008
The present invention relates to compounds of formula I ##STR00001## wherein R.sup.1, R.sup.2, R.sup.3, R.sup.4, and R.sup.5 are as defined in the specification. Compounds of the invention are active on the GABAB receptor and are useful for treating a variety of CNS disorders, includ
7375226 Bi- and tricyclic substituted phenyl methanones May 20, 2008
The present invention relates to compounds of formula IA ##STR00001## whereinR.sup.1, R.sup.2, R.sup.3, and n are as defined in the specification, and to pharmaceutically active acid addition salts thereof. The compounds of the invention are useful in the treatment of neurological an
7241761 Phenyl-piperazine methanone derivatives, substituted by heterocyclic groups July 10, 2007
The present invention relates to compounds of the general formula I ##STR00001## wherein R.sup.1 is the group ##STR00002## and R.sup.2, R', R'', R.sup.3, R.sup.4, R.sup.5, R.sup.6, R.sup.7, X.sup.1, X.sup.1', X.sup.2, and N are as defined in the specification. Compounds of the inve
7220744 Monocyclic substituted phenyl methanones May 22, 2007
The present invention relates to compounds of formula I ##STR00001## wherein R.sup.1, R.sup.2, X.sup.1, and X.sup.2 are as defined in the specification and to pharmaceutically acceptable acid addition salts thereof. Such compounds are inhibitors of the glycine transporter 1 (GlyT-1)










 
 
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