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Inventor: Fugner; Armin
Address: Gau-Algesheim, DE
No. of patents: 15
Patents:
| Patent Number |
Title Of Patent |
Date Issued |
| 6489365 |
Amidine derivatives, the preparation and use thereof as medicaments with Itb4 antagonistic effec |
December 3, 2002 |
| Compounds of the formula ##STR1##which is explained more fully in the specification, may be prepared by conventional methods and used therapeutically in conventional galenic preparations. |
| 6037377 |
Amidine derivatives, the preparation and use thereof as medicaments with LTB4 antagonistic effec |
March 14, 2000 |
| Compounds of the formula ##STR1## which is explained more fully in the specification, may be prepared by conventional methods and used therapeutically in conventional galenic preparations. |
| 5731332 |
Substituted benzamidine compounds which have useful pharmaceutical activity |
March 24, 1998 |
| Compounds of formula ##STR1## and their therapeutic use, inter alia, as LTB.sub.4 -antagonists. Exemplary compounds are:(Methoxycarbonyl-imino-{4'-[2-(2-propylphenoxy)-ethoxy]-biphenyl-4-yl}-meth yl)-amine;(Benzyloxycarbonyl-imino-{4'-[2-(2-propylphenoxy)-ethoxy]-biphenyl-4-yl}-me |
| 5686496 |
Chemical compound, the preparation thereof and its use in pharmaceutical compositions |
November 11, 1997 |
| The new compound of formula ##STR1## may be prepared by conventional methods and used therapeutically as an LTB.sub.4 -receptor antagonist. |
| 4720496 |
Pyridotriazoloquinazolines and triazolopyridoquinazolines useful as antiallergics |
January 19, 1988 |
| Compounds of the formula ##STR1## wherein (a)R.sub.1 is hydrogen, lower alkyl, lower alkoxy or 8-halo;R.sub.2 is hydrogen, lower alkyl, lower alkoxy or a fused benzene ring; andR.sub.3 and R.sub.4, together with each other, are --N.dbd.N--NH--; or(b)R.sub.1 and R.sub.2, together with each ot |
| 4686219 |
11-(Piperazin- or homopiperazin-1-yl)-5H-imidazo-(2,1-C)(1,4)benzodiazepines useful as anti- |
August 11, 1987 |
| Compounds of the formula ##STR1## wherein R.sub.1 and R.sub.2, which may be identical to or different from each other, are each hydrogen, fluorine, chlorine, bromine, trifluoromethyl, hydroxyl, nitro, amino, cyano, methylsulfonamido, alkyl of 1 to 4 carbon atoms, alkoxy of 1 to 3 |
| 4647563 |
Heterocyclic compounds |
March 3, 1987 |
| Compounds of the formula ##STR1## wherein Het is ##STR2## n is an integer from 1 to 4, inclusive, preferably 2 or 3, R.sub.1 is H or acyl,R.sub.2 is H, R.sub.1 O, --NHSO.sub.2 R.sub.7, --NHCOR.sub.8, --NHCONHR.sub.8, --NH--CH.sub.2 --C.sub.6 H.sub.4 --R.sub.9, --CH.sub.2 |
| 4581367 |
1-phenyl-2-(heterocyclyl-alkyl-amino)-ethanols |
April 8, 1986 |
| Compounds of the formula whereinHet is a heterocycle;n is an integer from 1 to 4, inclusive, preferably 2 or 3;R.sub.1 is H or acyl;R.sub.2 is H, R.sub.1 O, --NHSO.sub.2 R.sub.7, --NHCOR.sub.8, --NHCONHR.sub.8, --NH--CH.sub.2 --C.sub.6 H.sub.4 --R.sub.9, --CH.sub.2 OH, --CH.sub.2 SO.sub.2 R |
| 4558061 |
Bronchospasmolytic 1-(3-methanesulfonamido-4-hydroxyphenyl)-2-[(3-(4-acyl-aminophenyl)-imid a |
December 10, 1985 |
| Compounds of the formula ##STR1## wherein n is 1 or 2, R.sub.1 is hydrogen, --CO--R.sub.2 or --SO.sub.2 R.sub.3,R.sub.2 is hydrogen, alkyl of 1 to 4 carbon atoms, alkoxy of 1 to 4 carbon atoms or (alkyl of 1 to 4 carbon atoms)amino, andR.sub.3 is alkyl of 1 to 4 carbon atoms,and non- |
| 4503060 |
3-Imino-3H-dibenzo-[c,f]-imidazo-[1,5-a]azepine pharmaceuticals |
March 5, 1985 |
| Compounds of the formula ##STR1## wherein R.sub.1, R.sub.2, R.sub.3 and R.sub.4 are each hydrogen, halogen, alkyl of 1 to 6 carbon atoms or alkoxy of 1 to 6 carbon atoms;R.sub.5 is hydrogen, alkyl of 1 to 6 carbon atoms or alkenyl of 3 to 6 carbon atoms;R.sub.6 is alkyl of 1 to 6 car |
| 4460581 |
(1-Hydroxy-2-amino-alkyl)-substituted benzoxazinones and benzoxazolinones |
July 17, 1984 |
| Compounds of the formula ##STR1## wherein A is a single bond, ##STR2## R.sub.1 is --OH, --0--acyl, chlorine or hydrogen; R.sub.2 is hydrogen, methyl or ethyl;R.sub.3 is ##STR3## m is 2, 3 or 4; n is 1, 2 or 3;R.sub.4 is hydrogen or lower alkyl;R.sub.5 is hydrogen, lower a |
| 4378361 |
Heterocyclic compounds |
March 29, 1983 |
| Compounds of the formula ##STR1## wherein Het is ##STR2## n is an integer from 1 to 4, inclusive, preferably 2 or 3, R.sub.1 is H or acyl,R.sub.2 is H, R.sub.1 O, --NHSO.sub.2 R.sub.7, --NHCOR.sub.8, --NHCONHR.sub.8, --NH--CH.sub.2 --C.sub.6 H.sub.4 --R.sub.9, --CH.sub.2 |
| 4341778 |
3,1 Benzoxazin-2-ones and use thereof |
July 27, 1982 |
| The invention relates to compounds of general formula I ##STR1## (wherein R.sub.1 and R.sub.2, which may be the same or different, each represents a hydrogen atom or a (C.sub.1 -C.sub.4) alkyl group;R.sub.3 and R.sub.4, which may be the same or different, each represents a hydrogen, |
| 4332802 |
11-Oxo-11H-pyrido[2,1-b]quinazoline-2-carboxylic acid and salts thereof, antiallergic compositio |
June 1, 1982 |
| This invention relates to the novel compound 11-oxo-11H-pyrido[2,1-b]quinazoline-2-carboxylic acid of the formula ##STR1## and non-toxic, pharmacologically acceptable salts thereof, as well as to pharmaceutical composition containing these compounds as active ingredients, and met |
| 4313931 |
Fused dibenzo imidazolo compounds, compositions and use |
February 2, 1982 |
| This invention relates to a compound of the formula ##STR1## wherein R.sub.1, R.sub.2, R.sub.3, and R.sub.4, which may be the same or different, each represent a hydrogen or halogen atom or an alkyl or alkoxy group of from 1 to 6 carbon atoms;R.sub.5 and R.sub.6, which may be the sam |
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