| Patent Number |
Title Of Patent |
Date Issued |
| 4894221 |
Method of treating plaque using morpholine compounds |
January 16, 1990 |
| Novel morpholino compounds having the general formula ##STR1## wherein R.sub.1 is a straight or branched alkyl group containing 8 to 16 carbon atoms at the 2- or 3-position of the morpholino ring, and R.sub.2 is a straight or branched alkyl group containing 2 to 10 carbon atoms, |
| 4636382 |
Morpholino compounds and compositions |
January 13, 1987 |
| Novel morpholino compounds having the general formula ##STR1## wherein R.sub.1 is a straight or branched alkyl group containing 8 to 16 carbon atoms at the 2- or 3-position of the morpholino ring, and R.sub.2 is a straight or branched alkyl group containing 2 to 10 carbon atoms, |
| 4629620 |
Membrane-coated sustained-release tablets and method |
December 16, 1986 |
| A sustained-release coated pharmaceutical tablet comprising a drug-containing tablet and a coating or membrane surrounding the same, wherein the coating or membrane is water-insoluble and insoluble in gastrointestinal fluids and consists essentially of a terpolymer of polyvinylchlori |
| 4629619 |
Membrane-coated sustained-release tablets and method |
December 16, 1986 |
| A sustained-release coated pharmaceutical tablet comprising a drug-containing tablet and a coating or membrane surrounding the same, wherein the coating or membrane is water-insoluble and insoluble in gastrointestinal fluids and consists essentially of a terpolymer of polyvinylchlori |
| 4557925 |
Membrane-coated sustained-release tablets and method |
December 10, 1985 |
| A sustained-release coated pharmaceutical tablet comprising a drug-containing tablet and a coating or membrane surrounding the same, wherein the coating or membrane is water-insoluble and insoluble in gastrointestinal fluids and consists essentially of a terpolymer of polyvinylchlori |
| 4447433 |
Diphenylbutyl-piperazinecarboxamides to treat pain |
May 8, 1984 |
| Compounds having the general formula ##STR1## as herein defined and pharmaceutically acceptable acid addition salts thereof. Pharmaceutical compositions containing said compounds. Methods of treatment of humans and animals by such compounds and compositions. |
| 4385057 |
Diphenylbutyl-piperazinecarboxamides in pharmaceutical compositions and methods |
May 24, 1983 |
| Compounds having the general formula ##STR1## as herein defined and pharmaceutically acceptable acid addition salts thereof. Pharmaceutical compositions containing said compounds. Methods of treatment of humans and animals by such compounds and compositions. |
| 4366162 |
Aryl ethers of N-alkyl-piperidines and acid addition salts thereof |
December 28, 1982 |
| Aryl ethers of N-alkyl-piperdines having the formula ##STR1## wherein R.sub.1 represents hydrogen, halogen including F, Cl and Br, a lower alkanoyl group (e.g. alkanoyl of up to five carbon atoms), an alkenyl group (having three to five carbon atoms) or phenoxy, R.sub.2 represent |
| 4344952 |
Method of treating diarrhoea with gamma-piperidino-butyrophenones |
August 17, 1982 |
| A method of treating diarrhoea and promoting weight gain in mammals by administration of an effective amount of a compound selected from the group consisting of 4-fluoro-.gamma.-(4-alkylpiperidino)-butyrophenone of the formula ##STR1## wherein R is lower alkyl having 1 to 6 carbo |
| 4308387 |
Diphenylbutyl-piperzinecarboxamides |
December 29, 1981 |
| Compounds having the general formula ##STR1## as herein defined and pharmaceutically acceptable acid addition salts thereof. Pharmaceutical compositions containing said compounds. Methods of treatment of humans and animals by such compounds and compositions. |
| 4235875 |
Anticaries piperidino compounds |
November 25, 1980 |
| Novel alkyl 1-(hydroxyalkyl)piperidines and acid addition salts thereof, useful as inhibitors of dental plaque and therefore also useful against dental caries and periodontitis, are disclosed. Methods of making same, orally-acceptable compositions thereof, a method of treating therewith, |
| 4183933 |
Diarylbutyl octahydropyrazinopyrimidinones and methods of medical treatment using them |
January 15, 1980 |
| 2,3,4,7,8,9-Substituted octahydropyrazinopyrimidinones and acid addition salts thereof. A process for the preparation of said compounds. A pharmaceutical composition comprising such a compound and a conventional carrier. A process for the preparation of said composition. Method of me |
| 4144320 |
Aminoalcohols |
March 13, 1979 |
| Aminoalcohol compounds and acid addition salts thereof, useful in the prevention and treatment of dental caries and periodontitis, are disclosed. Methods of preparing said derivatives, orally acceptable compositions containing said compounds, and a method of treatment therewith are a |
| 4119711 |
Piperidino derivatives |
October 10, 1978 |
| Novel spiro 1-(hydroxyalkyl)-piperidino derivatives and acid addition salts thereof, useful in the prevention and treatment of dental caries and periodontitis, are disclosed. Methods of preparing said derivatives, orally acceptable compositions containing said compounds, and a method of |
| 4070473 |
Piperidino-butyrophenones |
January 24, 1978 |
| Novel gamma-(4-lower-alkyl-4-lower-alkoxypiperidino)-p-fluorobutyrophenones and acid addition salts thereof, useful as central depressants, e.g., neuroleptics (antipsychotics). Pharmaceutical compositions thereof and method of treating therewith. |
| 4024264 |
Diphenylbutylpiperidines |
May 17, 1977 |
| Novel 4,4-diphenylbutyl-1-(4-benzoyl-4-hydroxy or acyloxy)-piperidines and acid addition salts thereof, useful as central depressants, e.g., neuroleptics (anti-psychotics), are disclosed. Methods of making same, pharmaceutical compositions thereof, a method of treating therewith, and |
| 4021564 |
Neuroleptic piperidine compounds |
May 3, 1977 |
| Novel 1-substituted-4-aroyl-4-hydroxy and -4-acyloxypiperidines and acid addition salts thereof, useful as central nervous system depressants and neuroleptics with pronounced antipsychotic effects, are disclosed. Methods of making same, pharmaceutical compositions thereof, a method of tr |